In contrast, substances that bind directly to an enzyme's active site or the binding site of the endogenous ligand of a receptor are called orthosteric regulators or modulators. The site to which …

The meaning of ALLOSTERIC is of, relating to, undergoing, or being a change in the shape and activity of a protein (such as an enzyme) that results from combination with another substance at a point …

“Allosteric” was first introduced to mean the other site (i.e., a site distinct from the active or orthosteric site), an adjective for “regulation” to imply a regulatory outcome resulting from ligand binding at …

An allosteric or regulatory site is a place where the effectors bind and they may function as the allosteric activators or inhibitors. We can call effectors the modulators because they alter the enzyme’s …

Allosteric regulation is the regulation of an enzyme or other protein by binding an effector molecule at the protein's allosteric site (that is, a site other than the protein's active site).

In this article, we will learn about allosteric regulation, including allosteric inhibition and allosteric activation, and see examples.

Allosteric control, in enzymology, inhibition or activation of an enzyme by a small regulatory molecule that interacts at a site (allosteric site) other than the active site (at which catalytic activity occurs).

6 days ago · Allosteric sites are generally less conserved across related proteins than active sites, allowing a drug to target only one specific form of an enzyme. This specificity reduces the likelihood …

Nov 29, 2025 · What does it mean if something is allosteric? It refers to regulation of a protein's activity by a molecule binding to a site other than the active site. This guide explores allosteric …

Jan 23, 2024 · “Allosteric” was first introduced to mean the other site (i.e., a site distinct from the active or orthosteric site), an adjective for “regulation” to imply a regulatory outcome resulting from ligand …